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Found 5 of ec50 for PROTEASOME SUBUNIT BETA TYPE-7
having polymerids = 50006568 and
complexids = 50000077
TargetProteasome subunit beta type-7(Homo sapiens (Human))
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50010992(CHEMBL3259883)
Affinity DataEC50:  4.20E+3nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome in intact human Karpas 1106p cells assessed as substrate hydrolysis using Suc-LLVY-(D)-ami...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-7(Homo sapiens (Human))
Weill Cornell Medical College

Curated by ChEMBL
LigandPNGBDBM50010987(CHEMBL3259880)
Affinity DataEC50:  1.54E+4nMAssay Description:Inhibition of chymotrypsin-like activity of 26S proteasome in intact human Karpas 1106p cells assessed as substrate hydrolysis using Suc-LLVY-(D)-ami...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50518761(CHEMBL4573271)
Affinity DataEC50:  2.40E+4nMAssay Description:Stimulation of human 20S proteasome using 11 amino acid FRET peptide as substrate measured every 2 mins over 1 hr by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50054471((5Z,8Z)-Icosa-5,8,11,14-tetraenoic acid (4-hydroxy...)
Affinity DataEC50:  2.80E+4nMAssay Description:Stimulation of human 20S proteasome using 11 amino acid FRET peptide as substrate measured every 2 mins over 1 hr by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50518762(CHEMBL4561568)
Affinity DataEC50:  3.50E+4nMAssay Description:Stimulation of human 20S proteasome using 11 amino acid FRET peptide as substrate measured every 2 mins over 1 hr by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed